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Tocris/Nepicastat hydrochloride/5037/10/10 mg
  • Tocris/Nepicastat hydrochloride/5037/10/10 mg

Tocris/Nepicastat hydrochloride/5037/10/10 mg

价格: ¥1908.00 市场价: 3180.00

货号: 5037/10
品牌: Tocris
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    • Description:Potentandselectivedopamineβ-hydroxylase(DBH)inhibitor;orallybioavailable
      ChemicalName:5-(Aminomethyl)-1-[(2S)-5,7-difluoro-1,2,3,4-tetrahydro-2-naphthalenyl]-1,3-dihydro-2H-imidazole-2-thionehydrochloride
      Purity:≥98%(HPLC)
      BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

      BiologicalActivity

      Potentandselectivedopamineβ-hydroxylase(DBH)inhibitor(IC50=9nM).SelectiveforDBHover12otherenzymes.Decreasesnoradrenalineandincreasesdopaminelevelsintissuesandplasmainhypertensiverats.Preventsprogressiveleftventriculardysfunctioninaninvivoheartfailuremodel.Alsopotentiatesthestimuluseffectsofcocainewithoutproducingcocaine-likeeffectsinrats.Orallybioavailable.

      TechnicalData

      M.Wt331.81
      FormulaC14H15F2N3S.HCl
      StorageStoreat-20°C
      Purity≥98%(HPLC)
      CASNumber170151-24-3
      PubChemID9840545
      InChIKeyDIPDUAJWNBEVOY-PPHPATTJSA-N
      SmilesS=C(NC=C3CN)N3[C@H]2CCC1=C(F)C=C(F)C=C1C2.Cl

      Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

      AllTocrisproductsareintendedforlaboratoryresearchuseonly.

      SolubilityData

      SolventMaxConc.mg/mLMaxConc.mM
      Solubility
      DMSO33.18100

      PreparingStockSolutions

      Thefollowingdataisbasedontheproductmolecularweight331.81.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

      Concentration/SolventVolume/Mass1mg5mg10mg
      1mM3.01mL15.07mL30.14mL
      5mM0.6mL3.01mL6.03mL
      10mM0.3mL1.51mL3.01mL
      50mM0.06mL0.3mL0.6mL

      ProductDatasheets

      CertificateofAnalysis/ProductDatasheet
      SafetyDatasheet

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